Biomedical Engineering Reference
In-Depth Information
4-Aminopiperidine
VU0184670
mAChR M
1
agonist;
EC
50
=
Cell-based calcium flux
assay using Fluo-4
45
152 nM
Benzopyran-succinimide
analog
Androgen receptor
antagonist; 15.1% of full
activity at
10
M and 10
M DHT
Modified cell line
expressing androgen
receptor-binding
element and a luciferase
reporter
46
Benzopyran-maleimide
ampkinone
AMPK activator 322%
relative phosphorylation
activity at 10
M
Immunoblotting assay
detecting
phosphorylated AMPK
substrate
47
(
continued
)
