BREAST CANCER RESISTANCE PROTEIN - Drug Transporters: Molecular Characterization and Role in Drug Disposition - page 330

Substrates Inhibitors

Hesperetin 111
Daidzein 111
Resveratrol 111
Genistein 113
Naringenin-7-glucoside 113
Benzimidazoles
Pantoprazole 119
Omeprazole 119
Oxfendazole 195
Estrogens, estrogen agonists,
and estrogen antagonists

2-Amino-1-methyl-6-phenylimidazo(4,5- b )pyridine
(PhIP) 88 , 132 , 138
Porphyrins
Pheophorbide a 83 , 84
Pyropheophorbide, a methyl ester 85
Chlorin e6 85
Protoporphyrin IX 54 , 85
Fluorescent compounds
Rhodamine 123 a 8 , 44 , 79
Lysotracker Green a 44 , 79
BODIPY-prazosin 44 , 79
Hoechst 33342 82 , 189
Flavonoids
Genistein 113
Quercetin 97 , 190
Glucuronide, glutathione, and sulfate conjugates
Benzo[ a ]pyrene-3-sulfate (BP3S) 191
Benzo[ a ]pyrene-3-glucuronide (BP3S) 191
Estrone 3-sulfate 87 , 89 , 95
4-Methylumbelliferone sulfate 89
4-Methylumbelliferone glucuronide 140
6-Hydroxy-5,7-dimethyl-2-methylamino-4-
(3-pyridylmethyl)benzothiazole
glucuronide (E3040) 89 , 192
Dehydroepiandrosterone sulfate
(DHEAS) 192 , 193
17 -Estradiol sulfate 87
Acetaminophen sulfate 194
Benzimidazoles
Albendazole sulfoxide 195
Oxfendazole 195
Pantoprazole 119
Antibiotics
Ciprofloxacin 90
Ofloxacin 90
Norfloxacin 90
Erythromycin 91
Dirithromycin 91
Rifampicin 91
Nitrofurantoin 53
Dihydrotestosterone 196
Sulfasalazine 197 , 198
Phenethyl isothiocyanate 116 , 199
Dipyridamole 118
Ochratoxin A 200
GV196771 201
Folic acid 184
Cimetidine 88
ME3229 202

-Estradiol 105
Estrone 105
Diethylstilbestrol 106
Tamoxifen 106
Toremifene 106
TAG-11 106
TAG-139 106
Taxanes
Ortataxel a 120
tRA96023 a 120
tRA98006 a 122
Flavopiridol 68
UCN-01 83
Novobiocin a 205 , 206 , 206
Stilbenoids 207

17

a Compound affected by the amino acid at position 482.