Biomedical Engineering Reference
In-Depth Information
TABLE 18.1 ( Continued )
Structure
Name
Activity
Assay
Ref.
Dihydroquinolin-5-one
analog
Mycobacterium
tuberculosis (MTB)
inhibitor; MIC = 1.56
g/mL
Minimum inhibitory
concentration assay
15
Naphthoquinone analog
Cell migration inhibitor;
IC 50 = 14.8 M
Wound closure assay
with breast cancer cells
(MDA-MB-231)
16
N -Pyridin-2-yl
hydroxylamine analog
Antibacterial activity;
MIC 90 =
MIC assay using the
broth microdilution
method
17
M against
Micrococcus luteus
2
Synthetic sesquiterpene
analog
Antitrypanosomal
activity; IC 50 = 0.55
g/mL
Activity against
Trypanosoma brucei
18
 
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