Biomedical Engineering Reference
In-Depth Information
TABLE 18.1 (
Continued
)
Structure
Name
Activity
Assay
Ref.
Dihydroquinolin-5-one
analog
Mycobacterium
tuberculosis
(MTB)
inhibitor; MIC
=
1.56
g/mL
Minimum inhibitory
concentration assay
15
Naphthoquinone analog
Cell migration inhibitor;
IC
50
=
14.8
M
Wound closure assay
with breast cancer cells
(MDA-MB-231)
16
N
-Pyridin-2-yl
hydroxylamine analog
Antibacterial activity;
MIC
90
=
MIC assay using the
broth microdilution
method
17
M against
Micrococcus luteus
2
Synthetic sesquiterpene
analog
Antitrypanosomal
activity; IC
50
=
0.55
g/mL
Activity against
Trypanosoma brucei
18