Biomedical Engineering Reference
In-Depth Information
TABLE 18.1
( Continued )
Structure
Name
Activity
Assay
Ref.
Dihydropyrimidine
emmacin
Prokaryote-selective
dihydrofolate reductase
(DHFR) inhibitor; IC 50
= 5.4 M
EMRSA bacterial
proliferation phenotypic
assay
9
Homopiperidine
gemmacin
Cell
membrane-disrupting
antibiotic; MIC 50 =
Minimum inhibitory
concentration (MIC)
assay
10
8.0
g/mL against
EMRSA-15
Furochromane analog
Mycobacterium
tuberculosis (MTB)
inhibitor; MIC 95 = 0.6
g/mL
Microdilution resazurin
assay
11
 
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