Biomedical Engineering Reference
In-Depth Information
Hepatic CL int
In Vivo CL
NF54
Hepatic CL int
In Vivo CL
NF54
Compound
Mouse
Human
(mL/min/kg)
IC 50 (nM)
Compound
Mouse
Human
(mL/min/kg)
IC 50 (nM)
90
High
High
49.66
9
——
20
Low
Low
>
5000
SR - 25
——
> 5000
126
SR - 19
444
Low
Low
9.75
0.9
1808
Low
Low
2.58
77
SS - 25
SR - 27
 
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