Biomedical Engineering Reference
In-Depth Information
Acknowledgment
The author is grateful to Dagmar Stumpfe for review of the chapter and help with
illustrations.
REFERENCES
1. P. Ripphausen, B. Nisius, L. Peltason, J. Bajorath,
J. Med. Chem
.
2010
,
53
, 8461-8467.
2. D. Horvath,
J. Med. Chem
.
1997
,
40
, 2412-2423.
3. M. F. M. Engels, P. Venkatarangan,
Curr. Opin. Drug Discov. Dev
.
2001
,
4
, 275-283.
4. J. Bajorath,
Nat. Rev. Drug Discov
.
2002
,
1
, 882-894.
5. T. Polgar, G. M. Keseru,
Comb. Chem. High Throughput Screen
.
2011
,
14
, 889-897.
6. D. Stumpfe, P. Ripphausen, J. Bajorath,
Future Med. Chem
.
2012
,
4
, 593-602.
7. D. Stumpfe, J. Bajorath, in:
Methods and Principles in Medicinal Chemistry. Virtual
Screening. Principles, Challenges, and Practical Guidelines
, C. Sotriffer, Ed., Wiley-
VCH, Weinheim, Germany,
2011
, pp. 73-103.
8. P. Ripphausen, B. Nisius, J. Bajorath,
Drug Discov. Today
2011
,
16
, 372-376.
9. P. Ripphausen, D. Stumpfe, J. Bajorath,
Future Med. Chem
.
2012
,
4
, 603-613.
10. W. P. Walters, M. T. Stahl, M. A. Murcko,
Drug Discov. Today
1998
,
3
, 160-178.
11. T. Langer, R. D. Hoffmann,
Curr. Pharm. Des.
2001
,
7
, 509-527.
12. H. Xu, D. K. Agrafiotis,
Curr. Top. Med. Chem.
2002
,
2
, 1305-1320.
13. I. Muegge,
Mini Rev. Med. Chem
.
2008
,
8
, 927-933.
14. B. K. Shoichet,
Nature
2004
,
432
, 862-865.
15. D. B. Kitchen, H. Decornez, J. R. Furr, J. Bajorath,
Nat. Rev. Drug Discov
.
2004
,
3
,
935-949.
16. F. L. Stahura, J. Bajorath,
Curr. Pharm. Design
2005
,
11
, 1189-1202.
17. H. Geppert, M. Vogt, J. Bajorath,
J. Chem. Inf. Model
.
2010
,
50
, 205-216.
18. Y. Hu, D. Stumpfe, J. Bajorath,
J. Chem. Inf. Model
.
2011
,
51
, 1742-1753.
19. G. Schneider, W. Neidhart, T. Giller, G. Schmid,
Angew. Chem. Int. Ed
.
1999
,
38
,
2894-2896.
20. N. Brown, E. Jacoby,
Mini Rev. Med. Chem
.
2006
,
6
, 1217-1229.
21. R. Li, D. Stumpfe, M. Vogt, H. Geppert, J. Bajorath,
J. Chem. Inf. Model
.
2011
,
51
,
2507-2514.
22. M. Vogt, D. Stumpfe, H. Geppert, J. Bajorath,
J. Med. Chem
.
2010
,
53
, 5707-5715.
23. E. J. Gardiner, J. D. Holliday, C. O'Dowd, P. Willett,
Future Med. Chem
.
2011
,
3
,
405-414.
24. K. Heikamp, J. Bajorath,
J. Chem. Inf. Model
.
2011
,
51
, 2254-2265.
25. Y. Wang, H. Eckert, J. Bajorath,
ChemMedChem
2007
,
2
, 1037-1042.
26. Y. Wang, J. Bajorath,
J. Chem. Inf. Model
.
2008
,
48
, 75-84.
27. H. Eckert, J. Bajorath,
Drug Discov. Today
2007
,
12
, 225-233.
28. J. Bajorath,
J. Chem. Inf. Comput. Sci
.
2001
,
41
, 233-245.
29. J. S. Mason, A. C. Good, E. J. Martin,
Curr. Pharm. Design
2001
,
7
, 567-597.