Chemistry Reference
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Table 1 Iron salts-catalyzed transformations of persilylated D -glucopyranoside deriva-
tives 50 and 51.
PhCHO 3 equiv
Et 3 SiH 1.1 equiv
catalyst
OTMS
Ph
O
O
O
O
TMSO
TMSO
O
X
X
TMSO
HO
CH 2 Cl 2 /CH 3 CN: 4/1
0 °C to rt
1.5-2h
Ph
50
:X =
α
-OMe
52 :X = α -OMe
53
51
:X =
β
-SPh
:X =
-SPh
β
Entry
X
Catalyst
Mol%
Yield%
1
α-OMe
FeCl 3
6H 2 O
5
77
66 a
2
a-OMe
FeCl 3 6H 2 O
1
3
a-OMe
FeCl 3
5
75
- b
4
a-OMe
Fe(acac) 3
5
- b
5
a-OMe
(FeCl 3 ) 2 (TMEDA) 3
2.5
14 a,c
6
a-OMe
Fe(NO 3 ) 3 9H 2 O
5
- a,d
7
a-OMe
FeCl 2 4H 2 O
5
8
β-SPh
FeCl 3
6H 2 O
5
71
a Overnight reaction.
b
Starting material was recovered.
c The 4,6-O-benzylidene derivative was obtained in 68% yield.
d
CH 2 Cl 2 was used instead of CH 2 Cl 2 /CH 3 CN; only the 4,6-O-benzylidene derivative was
isolated in 53% yield. acac = acetylacetone; TMEDA = N,N,N 0 ,N 0 -tetramethylethylenediamine.
TMSO
TMSO
TMSO
O
50 : X = α -OMe
51
: X =
β
-SPh
X
TMSO
Ph
O O
O
Ph
O
O
Ph
tandem
catalysis a
then
additive(s)
OMe
Et 3 SiH
5 equiv
Ac 2 O
5 equiv
HO O
O
O
54
, 64%
O
HO
Ph
OMe
Ph
O
O
59 , 55% b
O
Ph
O
O
Ph
OMe
HO O
O
O
SPh
55
O
, 58%
C 15 H 31
HO
Ph
58
, 54% b
Ph
O O
O
O
Ph
O O
O
O
SPh
Ph
OMe
O
O
O
Ph
56
, 60%
O
57
, 60%
a see
Scheme 14 Three-step transformations catalyzed by iron( III ) chloride in one-pot.
Table 1; b simultaneous addition of 5 mol% more of FeCl 3 6H 2 O was required.
glycosyl acceptors (Scheme 14). Hence, terminal addition of acetic an-
hydride, palmitoyl chloride or pivaloyl anhydride afforded the orth-
ogonally protected monosaccharides 54-57 in good yields. Noteworthy, a
higher temperature was required to proceed with a sterically hindered
acylating reagent.
The combination of iron( III ) chloride with triethylsilane can also pro-
mote the regioselective 4,6-O-benzylidene ring opening. Our results
showed that the addition of an excess of the reducing reagent was re-
quired for completion. Accordingly, persilylated pyranoside 50, treated
 
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