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46. Chen, S.-H.; Farina, V.; Vyas, D. M.; Doyle, T. W.; Long, B. H.; Fairchild, C. Synthesis
and biological evaluation of C-13 amide-linked paclitaxl (taxol) analogues. J. Org.
Chem., 1996, 61: 2065-2070.
47. Hoemann, M. Z.; Vander Velde, D. G.; Aub´, J.; Georg, G. I.; Jayasinghe, L. R. Synthesis
of 13-epi-taxol via a transannular delivery of a borohydride reagent. J. Org. Chem., 1995,
60: 2918-2921.
48. Kelly, R. C.; Wicnienski, N. A.; Gebhard, I.; Qualls, S. J.; Han, F.; Dobrowolski, P. J.;
Nidy, E. G.; Johnson, R. A. 12,13-isobaccatin III. Taxane enol esters (12,13-isotaxanes).
J. Am. Chem. Soc., 1996, 118: 919-920.
49. Samaranayake, G.; Magri, N. F.; Jitrangsri, C.; Kingston, D. G. I. Modified taxols. 5.
Reaction of taxol with electrophilic reagents and preparation of a rearranged taxol
derivative with tubulin assembly activity. J. Org. Chem., 1991, 56: 5115-5119.
50. Chordia, M. D.; Kingston, D. G. I.; Hamel, E.; Lin, C. M.; Long, B. H.; Fairchild, C. A.;
Johnston, K. A.; Rose, W. C. Synthesis and biological activity of A-nor-paclitaxel
analogues. Bioorg. Med. Chem., 1997, 5: 941-947.
51. Chen, S.-H.; Fairchild, C.; Mamber, S. W.; Farina, V. Taxol structure-activity relation-
ships: synthesis and biological evaluation of 10-deoxytaxol. J. Org. Chem., 1993, 58:
2927-2928.
52. Harriman, G. C. B.; Jalluri, R. K.; Grunewald, G. L.; Vander Velde, D. G.; Georg, G. I.
The chemistry of the taxane diterpene: stereoselective synthesis of 10-deacetoxy-11,12-
epoxypaclitaxel. Tetrahedron Lett., 1994, 36: 8909-8912.
53. Marder, R.; Bricard, L.; Dubois, J.; Gu´nard, D.; Gu´ritte-Voegelein, F. Taxoids: 11,12-
dihydro-4-deacetyldocetaxel. Tetrahedron Lett., 1996, 37: 1777-1780.
54. Ojima, I.; Fenoglio, I.; Park, Y. H.; Sun, C.-M.; Appendino, G.; Pera, P.; Bernacki, R. J.
Synthesis and structure-activity relationships of novel nor-seco analogues of taxol and
taxotere. J. Org. Chem., 1994, 59: 515-517.
55. Ojima, I.; Lin, S.; Chakravarty, S.; Fenoglio, I.; Park, Y. H.; Sun, C. M.; Appendino, G.;
Pera, P.; Veith, J. M.; Bernacki, R. J. Syntheses and structure-activity relationships of
novel nor-seco taxoids. J. Org. Chem., 1998, 63: 1637-1645.
56. Appendino, G.; Belloro, E.; Grosso, E. D.; Minassi, A.; Bombardelli, E. Synthesis and
evaluation of 14-nor-A-secotaxoids. Eur. J. Org. Chem., 2002, 277-283.
57. Wang, M.; Xia, X.; Kim, Y.; Hwang, D.; Jansen, J. M.; Botta, M.; Liotta, D. C.; Snyder,
J. P. A unified and quantitative receptor model for the microtubule binding of paclitaxel
and epothilone. Org. Lett., 1999,1:43-46.
58. Nicoletti, M. I.; Colombo, T.; Rossi, C.; Monardo, C.; Stura, S.; Zucchetti, M.; Riva, A.;
Morazzoni, P.; Donati, M. B.; Bombardelli, E.; D'Incalci, M.; Giavazzi, R. IDN5109, a
taxane with oral bioavilabity and antitutmor acitivity. Cancer Res., 2000, 60: 842-846.
59. Huang, G. Y.; Guo, J. Y.; Liang, X. T. Studies on structure modificaton and structure-
activity relationship of new taxoids derived from sinenxan A. Acta Pharm. Sin., 1998,
33: 576-586.
60. Yin, D.; Liu, R.; Wang, D.; Guo, J.; Liang, X.; Sekiguchi, Y.; Kameo, K. Synthesis of
analogues of paclitaxel with 14b-side chain from sinenxan A. J. Chin. Pharm. Sci., 1999,
8: 191-196.
61. Liu, R. W.; Yin, D. L.; Wang, D. H.; Li, C.; Guo, J. Y.; Liang, X. T. Synthesis and
structure-activity relationships of novel 14b-side chain taxol derivatives. Acta Pharm.
Sin., 1998, 33: 910-918.
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