Carbohydrates in Peptide and Protein Design - Peptide and Protein Design for Biopharmaceutical Applications - page 200

[31] D. F. Veber, R. M. Freidinger, D. S. Perlow, W. J. Paleveda, F. W. Holly,
R. G. Strachan, R. F. Nutt, B. H. Arison, C. Homnick, W. C. Randall,
M. S. Glitzer, R. Saperstein and R. Hirschmann, A potent cyclic hexapeptide analog
of somatostatin, Nature , 292, 55-57 (1981).
[32] R. Hirschmann, L. Ducry and A. B. Smith, Development of an efficient, region- and
stereoselective route to libraries based on the b- D -glucose scaffold, J. Org. Chem ., 65,
8307-8316 (2000).
[33] V. Chanault, J. Lalot and P. V. Murphy, Synthesis of somatostatin mimetics based on
1-deoxy nojirimycin, ChemMedChem , 3, 1071-1076 (2008).
[34] S. A. W. Gruner, E. Locardi, E. Lohof and H. Kessler, Carbohydrate-based mimetics
in drug design: Sugar amino acids and carbohydrate scaffolds, Chem. Rev ., 102,
491-514 (2002).
[35] K. Heyns and H. Paulsen, Synthese der D -Glucosaminurons ¨ ure (2-amino-2-desoxy-
D -glucurons ¨ ure) und einige ihrer Derivate, Chem. Ber ., 88, 188-195 (1955).
[36] T. K. Chakraborty, S. Ghosh and S. Jayaprakash, Sugar amino acids and their uses in
designing bioactive molecules, Curr. Med. Chem ., 9, 421-435 (2002).
[37] T. K. Chakraborty, S. Jayaprakash and S. Ghosh, Sugar amino acids - Novel
peptidomimetics and their potential in combinatorial synthesis, Comb. Chem. High
Throughput Screen ., 5, 373-387 (2002).
[38] A. Dondoni and A. Marra, Methods for anomeric carbon-linked and fused sugar
amino acid synthesis: The gateway to artificial glycopeptides, Chem. Rev ., 100,
4395-4421 (2000).
[39] M. D. P. Risseuw, M. Overhand, G. W. J. Fleet and M. I. Simone, A compendium of
sugar amino acids (SAA): Scaffolds, peptide- and glycomimetics, Tetrahedron
Asymmetry 18, 2001-2010 (2007).
[40] R. M. van Well, L. Marinelli, C. Altona, K. Erkelens, G. Siegal, M. van Raaij,
A. L. Llamas-Saiz, H. Kessler, E. Novellino, A. Lavecchia, J. H. van Boom and
M. Overhand, Conformational analysis of furanoid e-sugar amino acids containing
cyclic peptides by NMR spectroscopy, molecular dynamics simulation, and X-ray
crystallography: Evidence for a novel turn structure, J. Am. Chem. Soc ., 125,
10822-10829 (2003).
[41] A. B. Smith, S. Sasho, B. A. Barwis, P. Sprengeler, J. Barbosa, R. Hirschmann and
B. S. Cooperman, Design and synthesis of a tetrahydropyran-based inhibitor of mam-
malian ribonucleotide reductase, Bioorg. Med. Chem. Lett ., 8, 3133-3136 (1998).
[42] M. J. Sofia, R. Hunter, T. Y. Chan, A. Vaughan, R. Dulina, H. Wang and D. Gange,
Carbohydrate-based small-molecule scaffolds for the construction of universal phar-
mocophore mapping libraries, J. Org. Chem ., 63, 2802-2803 (1998).
[43] A. A. Edwards, O. Ichihara, S. Murfin, R. Wilkes, M. Whittaker, D. J. Watkin and G.
W. J Fleet, Tetrahydrofuran-based amino acids as library scaffolds, J. Comb. Chem .,
6, 230-238 (2004).
[44] K. C. Nicolaou, H. Fl ¨ rke, M. G. Egan, T. Barth and V. A. Estevez, Carbanucleotides
and carbopeptoids - New carbohydrate oligomers, Tetrahedron Lett ., 36,

1775-1778 (1995).
[45] E. Locardi, M. St ¨ ckle, S. Gruner and H. Kessler, Cyclic homooligomers from sugar
amino acids: Synthesis, conformational analysis, and significance, J. Am. Chem. Soc .,
123, 8189-8196 (2001).
[46] B. A. Mayes, R. J. E. Stetz, W. G. Ansell and G. W. J. Fleet, Cyclo(6-amino-6-deoxy-
D -galactonic acid) 4 ,: a new class of carbopeptoid-cyclodextrins, Tetrahedron Lett .,
45, 153-156 (2004).